Synthesis and pharmacological characterization of Disila-AM80 (Disila-tamibarotene) and Disila-AM580, silicon analogues of the RARalpha-selective retinoid agonists AM80 (Tamibarotene) and AM580.
Reinhold Tacke
(1)
,
Volker Müller
(1)
,
Matthias W. Büttner
(1)
,
W Peter Lippert
(1)
,
Rüdiger Bertermann
(1)
,
Jürgen O. Daiss
(1)
,
Harshal Khanwalkar
(2)
,
Audrey Furst
(2)
,
Claudine Gaudon
(2)
,
Hinrich Gronemeyer
(2)