, Nature, vol.358, pp.15-16, 1992.
, Cold Spring Harbor Perspect. Biol, vol.9, pp.402-412, 1883.
, Annu. Rev.B iochem, vol.85, pp.3-75, 2016.
, Cell.S ignalling, vol.33, pp.49-58, 2017.
, Nature, vol.408, pp.7-310, 2000.
, Nat. CellB iol, vol.15, pp.49-53, 1991.
Cold Spring Harbor Perspect, Biol, vol.2, pp.1-17, 2010. ,
, J. Intern. Med, vol.277, pp.48-259, 2015.
, Nat. Rev.D rug Discovery, vol.13, pp.2243-2254, 2007.
, D. R. Carpizo, Mol. Pharmacol, vol.18, pp.67-575, 2012.
, J. Clin. Oncol, vol.30, pp.3633-3639, 2012.
, Cell Death Dis, vol.6, pp.1794-1804, 2015.
, Cell Death Dis, vol.4, pp.881-887, 2013.
, Metallomics, vol.2, pp.442-449, 2010.
, Proc. Natl.A cad.S ci. USA 2012, vol.109, pp.3590-13595
, Cancer Cell, vol.21, pp.6-14, 2012.
, Cell Cycle, vol.10, pp.1679-1689, 2011.
, Oncotarget, vol.5, pp.879-8892, 2014.
, Curr.Opin.C hem. Biol, vol.37, pp.26-32, 2017.
, Bioconjugate Chem, vol.59, pp.807-1812, 2016.
, Proc. Natl. Acad. Sci, vol.105, pp.360-10365, 2008.
, Proc. Natl. Acad. Sci, vol.11, pp.13584-13589, 2012.
, Neurotherapeutics, vol.245, pp.6-93, 2009.
, Prog. Neurobiol, vol.94, pp.47-359, 2011.
, Chem. Eur.J, vol.24, pp.17734-17742, 2018.
,
, , vol.48, pp.6-523, 2005.
, Chem. Sci, vol.8, pp.5636-5643, 2017.
, Neurotherapeutics, vol.6, pp.1-3, 2009.
, Neural Regener.Res, vol.7, pp.313-318, 2012.
, Mol. Pharmacol, vol.87, pp.825-831, 2015.
, Inorg. Chem, vol.48, pp.5928-5937, 2009.
, Drug Discovery Today, vol.20, pp.1391-1397, 2015.
, Biochemistry, vol.42, pp.2396-2403, 2003.
, A. R. Fersht, Proc. Natl.A cad.S ci, vol.94, pp.14338-14342, 1997.
, J. Am. Chem. Soc, vol.134, pp.6625-6636, 2012.
, Proc. Natl. Acad.S ci.U SA 2010, vol.107, pp.6097-6104, 1979.
, Coord. Chem. Rev, vol.184, pp.3-11, 1999.
, Cell. Calcium, vol.31, pp.245-251, 2002.
, Prostate, vol.68, pp.1443-1449, 2008.
CancerC hemother.P harmacol, J. Pharmacol. Exp. Ther, vol.8, pp.7280-7287, 2005. ,
, Nat. Rev.C ancer, vol.6, pp.813-823, 2006.
, Oncotarget, vol.4, pp.2186-2207, 2013.
, , vol.7, pp.1369-1378, 2007.
, Pharmaceutical Statistics, vol.10, pp.128-134, 2011.
Bevilacqua, A. Te sei, Drug Discovery Today, vol.18, pp.240-249, 2013. ,
, SLAS Discovery, vol.130, pp.1-17, 2007.
, Gastric Cancer, vol.20, pp.2663-2671, 2014.
, Nature, vol.407, pp.770-776, 2000.
, Oncotarget, vol.8, pp.1-5338, 2017.
, Br.J.Cancer, vol.91, pp.1931-1946, 2004.
, Proc. Natl. Acad.S ci. USA 2013, vol.110, pp.356-368, 2002.
, Mol. Cell. Biol, vol.21, pp.220-2225, 2001.
, Cancer Cell, vol.25, pp.304-317, 2014.
, Oncogene, vol.27, pp.6507-6521, 2008.
, Biochem.P harmacol, vol.71, pp.1540-1550, 2006.
6034 -6044;b)inSimilar reports by Fersht and co-workers show p53 Y220C-depedent induction of caspase-3 at 200 mm for PK7088, however,a ta ne arlier timep ointo f 6hours (seeR ef. [44a]). Boeckler and co-worker also reportN UGC3-depedent induction of apoptosis after 6h ours, Nucleic Acids Res, vol.41, 2013. ,
, Proc. Natl. Acad. Sci, vol.113, pp.5271-5280, 2016.
, Accepted manuscript online, 2018.
, Version of record online, 2018.
, Chem. Eur.J, vol.24, pp.17734-17742, 2018.
,