97–139: 27-O-3-(2-[3-carboxyacryloylamino]-5-hydroxyphenyl)-acryloyloxymyricerone
A127722: trans-trans-2-(4-methoxyphenyl)-4-(1,3-benzodioxol-5-yl)-1-([N,N-dibutylamino]carbonylmethyl)pyrrolidine-3-carboxylate
A81282: 4-(N-butyl-N-[{2′-(1H-tetrazol-5-yl)biphenyl-4-yl}methyl]amino)pyrimidine-5-carboxylic acid
A81988: 2-(N-n-propyl-N-[{2′-(1H-tetrazol-5-yl)biphenyl-4-yl}methyl]amino)pyridine-3-carbolic acid
antalarmin: N-butyl-N-ethyl-(2,5,6-trimethyl)-7-[2,4,6-trimethylphenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amine
BIBP3226: R-N2-(diphenylacetyl)-N-(4-hydroxyphenyl)methyl-argininamide
BIBS222: 2-n-butyl-1-(4-[6-carboxy-2,5-di-chlorbenzoylamino]-benzyl)-6-N-(methylaminocarbonyl)-n-pentylamino-benzimidazole
BIBS39: 4′-([2-n-butyl-6-cyclohexylaminocarbonylamino-benzimidazole-1-yl]-methyl)biphenyl-carboxylic acid
BMS180560: 2-butyl-1-chloro-1-([1-{2-(2H-tetrazol-5-yl)phenyl}-1H-indol-4-y]methyl)-1H-imidazole-5-carboxylic acid
BMS182874: 5-(dimethylamino)-N-(3,4-dimethyl-5-isoxazolyl)-1-naphthalenesulphonamide
BNTX: (5α)-17-(cyclopropylmethyl)-4,5-epoxy-3, 14-dihydroxy-7-(phenylmethylene)-morphinan-6-one hydrochloride
CAM4515: (S)-[1-(1H-indol-3-ylmethyl)-2-[methyl(phenylmethyl)amino]-2-oxoethyl]-2-benzofuranylmethyl ester, carbamic acid
CAM4750: [S-(R*,S*)]-[1-(1H-indol-3-ylmethyl)-1-methyl-2-[methyl[1-(4-pyridinyl)ethyl]amino]-2-oxoethyl]-2-benzofuranylmethyl ester monohydrochloride, carbamic acid
CGP49823: [(2R,4S)-2-benzyl-1-(3,5-dimethylbenzoyl)-N-[(4-quinolinyl)methyl]-4-piperineamine] dihydrocloride
CP122721: (+)-(2S,3S)-3-(2-methoxy-5-trifluoromethoxybenzyl)amino-2-phenylpiperidine
CP154526: butyl-ethyl-(2,5-dimethyl-7-[2,4,6-trimethylphenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino
CP96345: [(2S,3S)-cis-2-(diphenylmethyl)-N-(2-iodophenyl)-methyl]-1-azabicyclo-[2.2.2]octan-3-amino
CP99994: (+)-(2S,3S)-3-(2-methoxybenzylamino)-2-phenylpiperidine
CS866: (5-methyl-2-oxo-1,3-dioxolen-4-yl)methoxy-4-(1-hydroxy-1-methylethyl)-2-propyl-1-(4-[2-(tetrazol-5-yl)-phenyl]phenyl)methylimidazol-5-carboxylate
DMP811 (L708404): 4-ethyl-2-n-propyl-1-([2′-{1H-tetrazole-5-yl}biphenyl-4-yl]methyl)imidazole-5-carboxylic acid
DuP532: 2-propyl-4-pentafluorethyl-1-(2′-[2H-tetrazol-5-yl]-1,1′-biphenyl-4-yl-methyl)1H-imidazole-5-carboxylic acid
E4177: 4′-(2-cyclopropyl-7-methyl-3H-imidazo[5,4-b]pyridine-3-yl)methyl-2-biphenylcarboxylic acid
EXP3174: n-butyl-4-chloro-1-([2′-{1H-tetrazol-5yl}biphenyl-4-yl]methyl)imidazole-5-carboxylate
EXP3312: 2-n-propyl-4-chloro-1-[(2′-(1H-tetrazol-5-yl)biphenyl-4-yl)methyl]imidazole-5-carboxylaldehyde
EXP3892: 2-n-propyl-4-trifluoromethyl-1-[2′-(1H-tetrazol-5-yl)biphenyl-4-yl)methyl]imidazole-5-carboxilic acid
FK480: (S)-N-[1-(2-fluorophenyl)-3,4,6,7-tetrahydro-4-oxopyrrolo[3,2,1-jk][1,4]-benzodiazepine-3-yl]-1H-indole-2-carboxamide
FR173657: (E)-3-(6-acetamido-3-pyridyl)-N-(N-[2,4-dichloro-3{(2-methyl-8-quinolinyl)oxymethyl}phenyl]-N-methylaminocarbonyl-methyl)acrylamide
FR193108: (+)-3-[[5-(2-fluorophenyl)-9-methyl-2-oxo-3-[[[[3-(1H-tetrazol-5-yl)phenyl]amino]carbonyl]amino]-2,3-dihydro-1H-1,4--benzodiazepin-1-yl]acetyl]-3-azabicyclo[3.2.2]nonane
GR117289: 1-([3-bromo-2-[2-(1H-tetrazol-5-yl)phenyl]-5-benzofuranyl]methyl)-2-butyl-4-chloro-1H-imidazole-5-carboxylic acid
GR159897: 5-fluoryl-3-ylethyl(4-[phenylsulphinylmethyl])piperidine
GR203040: (+)-(2S,3S and 2R,2R)-2-methoxy-5-tetrazol-1-yl-benzyl-(2-phenyl-piperidin-3-yl)amine
GR205171: (2S-cis)-N-[[2-methoxy-5-[5-(trifluoromethyl)-1H-tetrazol-1-yl]phenyl]methyl]-2-phenyl-3-piperidinamine
GV150013: (+)-N-(1-[1-adamantane-1-methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-1H-1,5-benzodiazepin-3-yl)-N′-phenylurea
ICID6888: 2-ethyl-5,6,7,8-tetrahydro-4-([2′-{1H-tetrazol-5-yl}biphenyl-4-yl]methoxy)quinoline
ICID8731: 2-ethyl-4-([2′-{1H-tetrazol-5-yl}biphenyl-4-yl]methoxy)quinoline
KSG504: (S)-arginium(R)-4-[-N-(3-methoxypropyl)-N-pentylcarbamoyl]-5-(2-naphtylsulfonyl)pentanoate monohydrate
kuwanonH: [1S-(1a,5a,6b)]-8-[6-[2,4-dihydroxy-3-(3-methylbut-2-enyl)benzoyl]-5-(2,4-dihydroxyphenyl)-3-methylcyclohex-2-en-1-yl]-2-(2,4-dihydroxyphenyl)-5,7-dihydroxy-3-(3-methylbut-2-enyl)-4H-1-benzopyran-4-one
L158809: 5,7-dimethyl-2-ethyl-3-(2-[1H-tetrazol-5-yl]biphenyl-4-yl)lmidazol[4,5-b]pyridine
L161638: N-[2-ethyl-3-,4-dihydro-4-oxo-3-[[2′-(1H-tetrazol-5-yl)[1,1′-biphenyl]-4-yl]methyl]-6-quinazolinyl]-N-(phenylmethyl)-2-thiophenecarboxamide
L161664: 1-(N,N-diphenylaminocarbonyl)-4-(′N′,N′-di-n-pentylaminocarbonyl)piperazine-2-diethylaminopropylcarboxamide
L163017: 6-(benzoylamino)-7-methyl-2-propyl-3-([2′-{N-(3-methyl-1-butoxy)carbonylaminosulfonyl}(1,1′)-biphenyl-4-yl]methyl)-3H-imidazo(4,5-b)pyridine
L365031: 1-methyl-3-(4-bromobenzoyl)amino-5-phenyl-3H-1,4-benzodiazepin-2-one
L365260: 3R(+)-N-(2,3-dihydro-1-methyl-2-oxo-5-phenyl-1H-1,4-benzodiazepin-3-yl)-N′-(3-methylphenyl)urea
L367773: (1S,2S)-2,3-dihydro-1′-(((7,7-dimethyl-2-((4-imidazolylacetyl)amino)bicyclo[2.2.1]hept-1-yl)methyl)sulfonyl)spiro(1H-indene-1,4′-piperidine), hydrochloride
L368899: 1-([2-{2-amino-4-(methylsulphonyl)butyramido}-7,7-dimethylbicyclo[2.2.1]-heptan-1-yl]methylsulphonyl)-4-(2-methylphenyl)piperazine
L368935: N-(1,3-dihydro-1-(2-methyl)-propyl-2-oxo-5-phenyl-1H-1,4-benzodiazepin-3-yl)-N-([3-{1H-tetrazol-5-yl}phenyl]urea)
L371257: 1-(1-[4-{(N-acetyl-4-piperidinyl)oxy}-2-methoxybenzoyl]piperidinin-4-yl)-4H-3,1-benzoxazin-2-1H-one
L733060: (2S,3S)-3-([3,5-bis(trifluoromethyl)phenyl]methyloxy)-2-phenyl piperidine
L740093: N-([3R]-5-[3-azabicyclo{3.2.2}nonan-3-yl]-2,3-dihydro-1-methyl-2-oxo-1H-1,4-benzodiazepin-3-yl)-N′-(3-methylphenyl)urea
L742694: 2-(S)K[3,5-bis(trifluoromethyl)benzyl]oxy)-3-(S)-phenyl-4-(5-{3-oxo-1,2,4-triazolo}methylmorpholine
L743345: 3S-N-(3-azabicyclo[3.2.2.]nonan-3-yl-2,3-dihydro-1-methyl-2-oxo-1H-1,4-benzodiazepin-3-yl)-1H-indole-2-carboxamide
L749329: N-(2-[4-carboxy-2-propylphenoxy]-2-[dioxolo(e)phenyl]-acetyl)-(4-[1-methyl-ethyl)phenylsulfonylamide
L751281: dipotassium 4-(2-[1,3-benzodioxol-5-yl]-3-[4-isopropylphenylsulphonamido]-3-oxo-prop-1-yl)-3-propylbenzoate
L754142: dipotassium (−)-4-(1-[1,3-benzodioxol-5-yl]-2-[4-isopropylphenylsulphonamido]-2-oxoethoxy)-3-propylbenzoate
LR-B/081: methyl-2-([4-butyl-2-methyl-6-oxo-5-{[2′-(1H-tetrazol-5-yl)[1,1′-biphenyl]-4-yl]methyl}-1 (6H)-pyrimidinyl]methyl)-3-thiophenecarboxylate
LY191009: trans-5-(2-chlorophenyl)-3-oxo-4-phenyl-N-(4-[trifluoromethyl]phenylpyrazolidine-1-carboxamide
LY202769: 2-[2-(5-chloro-1H-indol-3-yl)ethyl]-3-[3-(1-methylethoxy)phenyl]-4(3H)-quinazolinone
LY242040: trans-3-oxo-4,5-diphenyl-N-(4-[trifluoromethyl]phenylpyrazolidine-1-carboxamide
LY247348: 2-[2-(1H-indol-3-yl)ethyl]-3-[3-(1-methylethoxy)phenyl]-4(3H)-quinazolinone
LY262684: trans-N-(4-bromophenyl)-4,5-bis(2-chlorophenyl)-3-oxopyrazolidine-1-carboxamide
LY262691: trans-N-(4-bromophenyl)-3-oxo-4,5-diphenyl-1-pyrazolidinecarboxamide
LY288513: (4S,5R)-N-(4-bromophenyl)-3-oxo-4,5-diphenyl-1-pyrrazolidinecarboxamide
LY303870: (R)-1-(N-[2-methoxybenzyl]acetylamino)-3-(1H-indol-3-yl)-2-(N-[2-{4-piperidin-1-yl}piperidin-1-yl}acetyl]amino)propane
LY306740: (R)-1-(N-[2-methoxybenzyl]acetylamino)-3-(1H-indol-3-yl)-2-(N-[2-{4-cyclohexylpiperazin-1-yl}acetyl]amino)propane
MDL105212A: [(R)-1-(2-[3-{3,4-dichlorophenyl}-1-{3,4,5-trimethoxybenzoyl}-pyrrolidin-3-yl]-ethyl-4- phenylpiperidine-4-carboxamide, hydrochloride
MEN10930: (S)-N-[1-[[[2-[methyl(phenylmethyl)amino]-1-(2-naphthalenylmethyl)-2-oxoethyl]amJno]carbonyl]cyclohexyl]-1H-jndole-3-carboxamide
MK966 (L159282): N-(4′-[{5,7-dimethyl-2-ethyl-3H-imidazo(4,5-b)pyridin-3-yl}methyl][1,1′-biphenyl]-2-yl)sulfonylbenzamide
NB127914: 2-methyl-4-(N-propyl-N-cyclopropanemethylamino)-5-chloro-6-(2,4,6-tri-trichloroanilino)pyrimidine
NTB: naltriben methasulfonate
OPC21268: 1-(1-[4-{3-acetylaminopropoxy}benzoyl]-4-piperidil)-3,4-dihydro-2-1H-quinolinone
OPC31260: 5-dimethylamino-1-(4-[2-methylbenzoylamino]benzoyl)-2,3,4,5-tetrahydro-1H-benzazepine
PD123177: 1-(4-amino-3-methylphenyl)methyl-3-(diphenylacetyl)-4,5,6,7-tetrahydro-1H-imidazol[4,5-c]pyridine-6-carboxylate
PD123319: (S)-1-(4-[dymethylamino]-3-methylphenyl)methyl-5-(diphenylacetyl)-4,5,67-tetrahydro-1H-imidazol[4,5-c]pyridine-6-carboxylate
PD134308 (CI988): 4-([2-{(3-[1H-indol-3-yl]-2-methyl-1 oxo-2-[{(tricyclo[3.3.1.13,7]dec-2-yloxy)carbonyl}amino]propyl)amino}-1-phenylethyl]amino)-4-oxo-(R-[R*R*])-butanoate-N-methyl-D-glucamine
PD135158: 4-([2-{(3-[1H-indol-3-yl]-2-methyl-1-oxo-2-[{(1.7.7-trimethyl-(bicyclo[2.2.1]hept-2-yl)oxy)carbonyl}amino]propyl)amino}-1-phenylethyl]amino)-4-oxo-[1S-1α.2β[S*(S*)]4α])-butanoate-N-(α-methyl-N-[{D-glucamine (bicyclo system 1S-endo)
PD140548: N-(α-methyl-N-[{tricyclo(3.3.1.13,7)dec-2-yloxy}carbonyl]-L-tryptophyl)-D-3-(phenylmethyl)-β-alanine
PD142898: benzenebutanic acid, β-([3-{1H-indol-3-yl}-2-methyl-2-[{[(2-methylcyclohexyl)oxy]carbonyl}amino]-1-oxopropyl]amino)-(1S-[1α{S*(R*)}-2β])
PD154075: [R-(R*S*)]-[1-(1H-indol-3-ylmethyl)-1-methyl-2-oxo-2-[(1-phenylethyl)amino]ethyl]-2- benzofuranylmethyl ester, carbamic acid
PD154804: 3-(1,3-benzodioxol-5-yl)-4-cyclohexylmethyl-5-hydroxy-5-(4-methoxyphenyl)-2,5-dihydrofuran-2-one
PD155080: 2-benzo(1,3)dioxol-5-yl-3-benzyl-4-(4-methoxyphenyl)-4-oxobut-2-enoate
PD156707: 2-benzo(1,3)dioxol-5-yl-4-(4-methoxyphenyl)-4-oxo-3-(3,4,5-trimethoxybenzyl)-but-2-enoate
PD159020: 3-(1,3-benzodioxol-5-yl)-1-(1,3-benzodioxol-5-ylmethyl)-5-methoxy-6-(phenylmethoxy)-1H-indole-2-carboxylic acid
PD159110: 3-(1,3-benzodioxol-5-yl)-1-(1,3-benzodioxol-5-ylmethyl)-6-propoxy-1H-indole-2-carboxylic acid
PD159433: 1-(1,3-benzodioxol-5-ylmethyl)-5,6-S-dimethoxy-3-[3,4,5- trimethoxyphenyl)thio]-lH--indole-2-carboxylic acid
PD161182: [S-(R*,S*)]-[2-(2,3-difluropheyl)-1-{(7-ureidoheptyl)carbamoyl}ethyl}carbamic acid-2-methyl-1-phenylpropyl ester
PD165929: (S)-α-[[[[2,6-bis(1-methylethyl)phenyl]amino]carbonyl]amino]-α-methyl-N-[[1-(2-pyridinyl)cyclohexyl]methyl]-1H-indole-3-propanamide
Ro462005: 4-tert-butyl-N-(6-[2-hydroxyetoxy]-5-[3-methoxyphenoxy]-4-pyrimidinyl)-benzenesulphonamide
Ro468443: (R)-4-tert-butyl-N-(6-[2,3-dihydroxypropoxy]-5-[2-methoxyphenoxy]-2-[4-methoxyphenyl]-pyrimidin-4-yl)-benzenesulphonamide
RP67580: (1–imino-2-[2-methoxyphenyl]ethyl)-7,7-diphenyl-4-perhydroisoindolone (3αR,7αR)
RP69758: 3-(3-[N-{N-methyl-N-phenyl-carbamoylmethyl}-N-phenyl-carbamoylmethyl]ureido)phenylacetic acid
RP71483: (E)-2-(3-[3-hydroxyiminomethyl-phenyl]ureido)-N-(8-quinolyl)-N-([1,2,3,4-tetrahydro-1-quinolyl]carbonylmethyl)acetamide
RP72540: (RS)-2-(3-[3-{N-(3-methoxyphenyl)-N-(N-methyl-N-phenyl-carbamoylmethyl)carbamoylmethyl}ureido]phenyl)propionic acid
RP73870: (RS)-([{N-(3-methoxyphenyl)-N-(N-methyl-N-phenyl-carbamoylmethyl)carbamoylmethyl}-3- ureido]-3-phenyl)-2-ethylsulfonate, potassium salt
RPR100893: (3nS,4S,7aS)-7,7-diphenyl-4-(2-methoxyphenyl)-2-[(S)-2-(2-methoxyphenyl)propionyl]perhydroisoindol-4-ol
SB209598: 3-(2-carboxymethoxy-4-methoxyphenyl)-1-(6-chloro-1,3-benzodioxol-5-ylmethyl)-indole-2-carboxilic acid
SB209670: (+)-1S,2R,S-3-(2-carboxymethoxy-4-methoxyphenyl)-1-(3,4-methylenedioxyphenyl)-5-prop-1-yloxyindane-2-carboxylic acid
SB217242: 1S,2R,3S-3-(2-hydroxyethoxy-4-methoxyphenyl)-1-(3,4-methylenedioxyphenyl)-5-propoxyindane-2-carboxylic acid
SB223412: (S)-(-)-N-(α-ethylbenzyl)-3-hydroxy-2-phenylquinoline-4-carboxamide
SC51316: 5-([3,5-dibutyl-1H-1,2,4-trizol-1-yl]methyl)-2-(2-[1H-tetrazol-5-ylphenyl])pyridine
SC51895: 1,4-dibutyl-1,3-dihydro-3-([2′-{1H-tetrazol-5-yl}[1,1′-biphenyl]-4-yl]methyl)-2H-imidazol-2-one
SC52458: 2,5-dibutyl-2,4-dihydro-4-([2-{1H-tetrazol-5-yl}[1,1′-biphenyl]-4′-yl]methyl)-3H-1,2,4-triazol-3-one
SKF108566: (E)-α-([2-butyl-1 -{(4-carboxyphenyl)methyl}-1H-imidazol-5-yl]methylene)-2-thiophenepropanoate
SR 48692: 2-([1-{7-chloro-4-quinolinyl}-5-{2,6-dimethoxyphenyl}-1H-pyrazol-3-carbonyl]amino)adamantane-2-carboxylic acid
SR120107A: (R,R)-1-(2-[2-{2-naphtylsulphamoyl}-3-phenyl-propionamido]-3-[4-{N-(4-[dimethylaminomethyl]-cis-cyclohexylmethyl)amidino}phenyljpropionyl)-pyrrolidine
SR120819A: (R,R)-1-(2-[2-{2-naphtylsulphamoyl}-3-phenyl-propionamido]-3-[4-{N-(4-[dimethylaminomethyl]-trans-cyclohexylmethyl)amidino}phenyl]propionyl)-pyrrolidine
SR140333: (S)-1-(2-[3-{3,4-dichlorophenyl}-1-{3-isopropoxyphenylacetyl}piperidin-3-yl]ethyl)-4-phenyl-1-azoniabicyclo(2.2.2)octane chloride
SR142801: (S)-(N)-(1-[3-{1-benzoyl-3-(3,4-dichlorophenyl)piperidin-3-yl}propyl]-4-phenylpiperidin-4-yl)-N-methylacetamide
SR142948A: 2-([5-{2,6-dimethoxyphenyl}-1-{4-(N-[3-dimethylaminopropyl]-N-methylcarbamoy-2-isopropylphenyl}-1H-pyrazol-3-carbonyl]amino)adamantane-2-carboxylic acid, hydrochloride
SR27897: 1-([2-{4-(2-chlorophenyl)thiazole-2-yl}aminocarbonyl]indolyl)acetic acid
SR48968: (S)-N-methyl-N-(4-acetylamino-4-phenylpiperidino)-2-(3,4-dichlorophenyl)butylbenzamide
SR49059: (2S)-1 -([2R,3S]-[5-chloro-3-{chlorophenyl}-1-{3,4-dimethoxysulphonyl}-3-hydroxy-2,3-dihydro-1H-indole-2-carbonyl]-pyrrolidine-2-carboxamide)
T0632: sodium (S)-3-(1-[2-fluorophenyl]-2,3-dihydro-3-[{3-isoquinolinyl}-carbonyl]amino-6-methoxy-2-oxo-1H-indole)propanoate
TBC11251: N-(4-chloro-3-methyl-5-isoxazolyl)-2-[2-(6-methyl1,3-benzodioxol-5-yl)-1-oxoethyl]-thiopentene-3-sulphonamide
UP269-6: 5-methyl-7-propyl-8(-)[2′-(1H-tetrazol-5-yl)biphenyl-4-yl)methyl]-1,2,4-triazolo]1,5-c]pyrimidin-2(3H)-one
UR7198: rel-(1R*,2R*)-3-[[4-(2-carboxy-1-phenylpropyl)phenyl]methyl]-5,7-dimethyl-2-ethyl-3H-imidazol[4,5-b]pyridine
UR7280:3-tert-butyl-1-propyl-5-([2′-{1H-tetrazol-5-yl}-1,1′-biphenyl-4-yl]methyl)-1H-pyrazole-4-carboxylic acid
WIN 64338: ([4-{(2-[{bis(cyclohexylamino)methylene}amino]-3-[2-naphthyl]-1-oxopropyl)amino}phenyl]methyl)tributylphosphonium chloride monohydrochloride
WIN51708:17β-hydroxy-17α-ethynyl-5α-androstanol[3,2-b]pyrimido[1,2-a]benzimidazole
WIN62577:[1R-(1α,3aβ,3bα,15aα,15bβ17aα)]-1ethynyl-2,3,3a,3b,4,5,15,15a,15b,16,17,17a-dodecahydro-15a, 17a-dimethyl-1H-benzimidazo[2,1-b]cyclopenta[5,6]naphto[1,2-g]quinazolin-1-ol
XR510:1-([2′-{[(isopentoxycarbonyl)amino]sulfonyl}-3-fluoro(1,1′-biphenyl)-4-yl]methyl)-5-(3-[N-pyridin-3-ylbutanamido]propanoyl)-4-ethyl-2-propyl-1H-imidazole, potassium salt
YF476: (3R)-N-(1-[tert-butylcarbonylmethyl]-2,3-dihydro-2-oxo-5-[2-pyridil]-1H-1,4-benzodiazepin-3-yl)-N′-(3-[methylamino]phenyl)urea
YM022: (R)-1-(2,3-dihydro-1-[2′-methylphenacyl]-2-oxo-5-phenyl-1H-1,4-benzodiazepin-3-yl)-3-(3-methylphenyl)urea
YM087: 4′-(2-methyl-1,4,5,6-tetrahydroimidazo{4,5-d}{1}benzazepin-6-yl]carbonyl)-2-phenylbenzanilide monohydrocloride